PubMed (MeSH Keyword) for id: 53378764

Year	Number of Results
2011	1
2013	1
2014	3
2016	1
2017	3
2018	4
2024	0

1

Modulation of Heat Shock Response Proteins by ASS234, Targeted for Neurodegenerative Diseases Therapy.

Ramos E, Romero A, Marco-Contelles J, López-Muñoz F, Del Pino J. Ramos E, et al. Chem Res Toxicol. 2018 Sep 17;31(9):839-842. doi: 10.1021/acs.chemrestox.8b00192. Epub 2018 Aug 27. Chem Res Toxicol. 2018. PMID: 30133257

2

Neuroinflammation Signaling Modulated by ASS234, a Multitarget Small Molecule for Alzheimer's Disease Therapy.

Del Pino J, Marco-Contelles J, López-Muñoz F, Romero A, Ramos E. Del Pino J, et al. ACS Chem Neurosci. 2018 Dec 19;9(12):2880-2885. doi: 10.1021/acschemneuro.8b00203. Epub 2018 Jul 30. ACS Chem Neurosci. 2018. PMID: 30048111

3

Contilisant, a Tetratarget Small Molecule for Alzheimer's Disease Therapy Combining Cholinesterase, Monoamine Oxidase Inhibition, and H3R Antagonism with S1R Agonism Profile.

Bautista-Aguilera ÓM, Budni J, Mina F, Medeiros EB, Deuther-Conrad W, Entrena JM, Moraleda I, Iriepa I, López-Muñoz F, Marco-Contelles J. Bautista-Aguilera ÓM, et al. J Med Chem. 2018 Aug 9;61(15):6937-6943. doi: 10.1021/acs.jmedchem.8b00848. Epub 2018 Jul 18. J Med Chem. 2018. PMID: 29969030

4

In silico assessment of the metabolism and its safety significance of multitarget propargylamine ASS234.

Ramos E, Marco-Contelles J, López-Muñoz F, Romero A. Ramos E, et al. CNS Neurosci Ther. 2018 Oct;24(10):981-983. doi: 10.1111/cns.12990. Epub 2018 May 28. CNS Neurosci Ther. 2018. PMID: 29808538 Free PMC article. No abstract available.

5

Multitarget-Directed Ligands Combining Cholinesterase and Monoamine Oxidase Inhibition with Histamine H₃ R Antagonism for Neurodegenerative Diseases.

Bautista-Aguilera ÓM, Hagenow S, Palomino-Antolin A, Farré-Alins V, Ismaili L, Joffrin PL, Jimeno ML, Soukup O, Janočková J, Kalinowsky L, Proschak E, Iriepa I, Moraleda I, Schwed JS, Romero Martínez A, López-Muñoz F, Chioua M, Egea J, Ramsay RR, Marco-Contelles J, Stark H. Bautista-Aguilera ÓM, et al. Angew Chem Int Ed Engl. 2017 Oct 2;56(41):12765-12769. doi: 10.1002/anie.201706072. Epub 2017 Sep 1. Angew Chem Int Ed Engl. 2017. PMID: 28861918

6

In-vitro and in-vivo evaluation of the modulatory effects of the multitarget compound ASS234 on the monoaminergic system.

Esteban G, Van Schoors J, Sun P, Van Eeckhaut A, Marco-Contelles J, Smolders I, Unzeta M. Esteban G, et al. J Pharm Pharmacol. 2017 Mar;69(3):314-324. doi: 10.1111/jphp.12697. Epub 2017 Jan 30. J Pharm Pharmacol. 2017. PMID: 28134992

7

The proof-of-concept of ASS234: Peripherally administered ASS234 enters the central nervous system and reduces pathology in a male mouse model of Alzheimer disease.

Serrano MP, Herrero-Labrador R, Futch HS, Serrano J, Romero A, Fernandez AP, Samadi A, Unzeta M, Marco-Contelles J, Martínez-Murillo R. Serrano MP, et al. J Psychiatry Neurosci. 2017 Jan;42(1):59-69. doi: 10.1503/jpn.150209. J Psychiatry Neurosci. 2017. PMID: 27636528 Free PMC article.

8

Upregulation of Antioxidant Enzymes by ASS234, a Multitarget Directed Propargylamine for Alzheimer's Disease Therapy.

Ramos E, Romero A, Marco-Contelles J, Del Pino J. Ramos E, et al. CNS Neurosci Ther. 2016 Sep;22(9):799-802. doi: 10.1111/cns.12590. Epub 2016 Jul 6. CNS Neurosci Ther. 2016. PMID: 27380946 Free PMC article. No abstract available.

9

Wnt signaling pathway, a potential target for Alzheimer's disease treatment, is activated by a novel multitarget compound ASS234.

del Pino J, Ramos E, Aguilera OM, Marco-Contelles J, Romero A. del Pino J, et al. CNS Neurosci Ther. 2014 Jun;20(6):568-70. doi: 10.1111/cns.12269. Epub 2014 Apr 8. CNS Neurosci Ther. 2014. PMID: 24712554 Free PMC article. No abstract available.

10

Kinetic and structural analysis of the irreversible inhibition of human monoamine oxidases by ASS234, a multi-target compound designed for use in Alzheimer's disease.

Esteban G, Allan J, Samadi A, Mattevi A, Unzeta M, Marco-Contelles J, Binda C, Ramsay RR. Esteban G, et al. Biochim Biophys Acta. 2014 Jun;1844(6):1104-10. doi: 10.1016/j.bbapap.2014.03.006. Epub 2014 Mar 16. Biochim Biophys Acta. 2014. PMID: 24642166

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