Warning: The NCBI web site requires JavaScript to function. more...
An official website of the United States government
The .gov means it's official. Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you're on a federal government site.
The site is secure. The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.
Agonist activity at human PPARG in an in vitro cell free assay measured by time-resolved fluorescence resonance energy transfer method
Assay data:4 Active, 5 Activity ≤ 1 µM, 238 Tested
SummaryRelated BioAssays by Target
Compound was evaluated for inhibition of human ABCB11 in an in vitro assay with cellular components measured by filtration, liquid scintillation counting
Assay data:43 Active, 3 Activity ≤ 1 µM, 508 Tested
Binding affinity to PPARgamma (unknown origin)
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Agonist activity at GAL4-fused human PPARgamma expressed in HepG2 cells
Agonist activity at human PPARgamma transfected in HEK293 cells assessed increase in luciferase activity incubated for 24 hrs
Displacement of [3H]rosiglitazone from human PPAR-gamma incubated for 1 day by radioligand binding assay
Assay data:5 Active, 2 Activity ≤ 1 µM, 7 Tested
Agonist activity at PPAR-gamma in human BMMSC cells assessed as induction of adiponectin production in presence of IDX adipogenic induction medium and measured on day 5 by ELISA
Assay data:4 Active, 2 Activity ≤ 1 µM, 8 Tested
Inhibition of recombinant human MAO-B
Assay data:19 Active, 8 Activity ≤ 1 µM, 25 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Agonist activity at yeast Gal4-fused human PPARgamma transfected in human HepG2 cells assessed as transactivation by measuring beta-galactosidase activity incubated for 20 hrs by luminometry
Assay data:10 Active, 1 Activity ≤ 1 µM, 26 Tested
Agonist activity at human PPARgamma expressed in HEK293 cells by luciferase/beta-galactosidase reporter gene assay
Assay data:6 Active, 2 Activity ≤ 1 µM, 14 Tested
Agonist activity at pBIND tagged human PPARgamma expressed in human HEK293 cells incubated for 18 hrs by dual luciferase reporter assay relative to control
Assay data:1 Active, 1 Activity ≤ 1 µM, 4 Tested
Agonist activity at human PPARgamma measured by dual luciferase reporter gene assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 13 Tested
Partial agonist activity at PPARgamma LBD (unknown origin) assessed as increase in FITC-labeled PGC-1alpha coactivator peptide recruitment by HTRF assay
Assay data:4 Active, 3 Activity ≤ 1 µM, 4 Tested
Stabilization of PPARgamma LBD (unknown origin)/FITC-labeled PGC-1alpha (unknown origin) protein-protein interaction assessed as dissociation constant by fluorescence anisotropy assay
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
Partial agonist activity at sGSF-PPARgamma (unknown origin) assessed as CBP-1 recruitment by HT-FRET assay
Assay data:5 Active, 5 Activity ≤ 1 µM, 5 Tested
Agonist activity at Gal4-fused PPARgamma (unknown origin) expressed in human U2OS cells co-transfected with pSG5 expression vector preincubated for 40 hrs followed by substrate addition by microplate reader assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 2 Tested
Binding affinity to PPARgamma (unknown origin) by lanthascreen TR-FRET assay
Assay data:3 Active, 3 Activity ≤ 1 µM, 3 Tested
Agonist activity at PPARgamma (unknown origin)
Assay data:33 Active, 5 Activity ≤ 1 µM, 47 Tested
Agonist activity at recombinant N-terminal His6 -tagged GFP fused PPARgamma LBD (unknown origin) (203 to 477 residues) expressed in Escherichia cell Rosetta2 using biotinylated NLVPDAASKHKQLSELLRGGSGS peptide as substrate assessed as induction of Tb cryptate labelled CBP recruitment measured after 2 hrs by HTRF assay
Assay data:3 Active, 2 Activity ≤ 1 µM, 3 Tested
Agonist activity at human PPARgamma transfected in COS-7 cells assessed luciferase activity measured after 24 hrs by cell based luciferase transactivation assay
Assay data:4 Active, 1 Activity ≤ 1 µM, 10 Tested
Filters: Manage Filters
Your browsing activity is empty.
Activity recording is turned off.
Turn recording back on