BioAssays, Active for PubChem Compound (Select 126648559) - PubChem BioAssay - NCBI

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Select item 18275111.

Inhibition of BRD3-BD2 (unknown origin) assessed as dissociation constant by TR-FRET method

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 3

Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested

AID:: 1827511

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 18275102.

Inhibition of BRD3-BD1 (unknown origin) assessed as dissociation constant by TR-FRET method

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 3

Assay data:2 Active, 2 Tested

AID:: 1827510

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 17881213.

LPS-PBMC assay (MCP-1)

Source:: ChEMBL

Protein Target:: C-C motif chemokine 2

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1788121

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 17881204.

In vitro inhibition of MCP-1 in Lipopolysaccharide-stimulated human whole blood

Source:: ChEMBL

Protein Target:: C-C motif chemokine 2

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1788120

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 17881195.

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 4

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1788119

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 17881176.

BRDT BD2 Bromoscan (DiscoverX)

Source:: ChEMBL

Protein Target:: Bromodomain testis-specific protein

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1788117

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 17881157.

BRD4 BD2 Bromoscan (DiscoverX)

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 4

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1788115

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 17881138.

BRD3 BD2 Bromoscan (DiscoverX)

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 3

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1788113

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 17881119.

BRD2 BD2 Bromoscan (DiscoverX)

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 2

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1788111

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 178810910.

BET mutant TR-FRET assay (BRDT BD2)

Source:: ChEMBL

Protein Target:: Bromodomain testis-specific protein

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1788109

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 178810711.

BET mutant TR-FRET assay (BRD4 BD2)

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 4

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1788107

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 178810512.

BET mutant TR-FRET assay (BRD3 BD2)

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 3

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1788105

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 178810313.

BET mutant TR-FRET assay (BRD2 BD2)

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 2

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1788103

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 178804114.

TR-FRET assay (BRDT BD2)

Source:: ChEMBL

Protein Target:: Bromodomain testis-specific protein

Assay data:2 Active, 2 Activity ≤ 1 µM, 3 Tested

AID:: 1788041

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 178803915.

TR-FRET assay (BRD4 BD2)

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 4

Assay data:2 Active, 2 Activity ≤ 1 µM, 3 Tested

AID:: 1788039

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 178803716.

TR-FRET assay (BRD3 BD2)

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 3

Assay data:2 Active, 2 Activity ≤ 1 µM, 3 Tested

AID:: 1788037

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 178803517.

TR-FRET assay (BRD2 BD2)

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 2

Assay data:2 Active, 2 Activity ≤ 1 µM, 3 Tested

AID:: 1788035

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 177713818.

Inhibition of 6His-Thr-BRD4 (1 to 477 residues) BD1 domain (unknown origin) incubated for 30 mins by TR-FRET assay

Source:: ChEMBL

Protein Target:: Bromodomain-containing protein 4

Assay data:11 Active, 2 Activity ≤ 1 µM, 40 Tested

AID:: 1777138

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 177705619.

Binding affinity to 6His-Thr-BRD4 (1 to 477 residues) BD2 domain Y390A mutant (unknown origin) incubated for 30 mins by TR-FRET assay

Source:: ChEMBL

Assay data:48 Active, 47 Activity ≤ 1 µM, 49 Tested

AID:: 1777056

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation

Select item 177560520.

Inhibition of 6His-Thr-BRD4 (1 to 477 residues) BD2 domain Y390A mutant (unknown origin) incubated for 30 mins by TR-FRET assay

Source:: ChEMBL

Assay data:48 Active, 41 Activity ≤ 1 µM, 51 Tested

AID:: 1775605

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation

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BioActivity

Active Compounds (27)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 µM (26)
BioAssays with the active concentration of tested reagents less than 1 micromolar

Experiment Type

Confirmatory (27)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations

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Literature Extraction (12)
BioAssays extracted from the literature
Other (15)
BioAssays deposited by other experimentalists

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