Warning: The NCBI web site requires JavaScript to function. more...
An official website of the United States government
The .gov means it's official. Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you're on a federal government site.
The site is secure. The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.
Selectivity interaction (KinomScan Ambit) EUB0000622a MYLK
Assay data:1 Tested
SummaryRelated BioAssays by Target
Inhibition of MYLK in HEK293 cells by NanoBRET assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
MYLK DiscoveRx kinase panel
Inhibition of MYLK (unknown origin) at 1 uM by kinome scan method
Kinome Profiling from Article 10.1021/cb400407c: "Fluorescence Linked Enzyme Chemoproteomic Strategy for Discovery of a Potent and Selective DAPK1 and ZIPK Inhibitor."
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
MYLK/MLCK Assay from US Patent US10150755: "ASK1 inhibitor compounds and uses thereof"
Assay data:18 Active, 14 Activity ≤ 1 µM, 18 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Assay data:14 Active, 8 Activity ≤ 1 µM, 18 Tested
cGPK assay from Article 10.1016/0960-894X(94)00458-R: "Novel Indolocarbazole protein kinase C inhibitors with improved biochemical and physicochemical properties."
Assay data:20 Active, 15 Activity ≤ 1 µM, 21 Tested
KinomeScan assay: inhibition of MYLK
Assay data:108 Tested
smMLCK(MYL1LGF1) Takeda global kinase panel
Assay data:1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, activity ≤ 1 µMRelated BioAssays by Target
MYLK ProQinase selectivity panel
MYLK (MLCK) Kinase screen
MYLK Invitrogen selectivity data (BI)
myosin light chain kinase Millipore kinase panel
SMMLCK DUNDEE kinase screen (BI)
MYLK Invitrogen Lab (UK) kinase screen (BI)
MYLK(smMLCK) Kinase panel
Inhibition of MYLK (unknown origin) assessed as residual activity measured at 1 uM
Assay data:3 Tested
Filters: Manage Filters
Your browsing activity is empty.
Activity recording is turned off.
Turn recording back on