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Inhibition of KDM5A (unknown origin ) by TR-FRET assay
Assay data:3 Active, 2 Activity ≤ 1 µM, 3 Tested
SummaryRelated BioAssays by Target
Inhibition of Halo-tagged KDM5A PHD3 domain (unknown origin)
Assay data:3 Tested
Inhibition of KDM5A (unknown origin ) demethylase activity using H3 as substrate by Chemiluminescent assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Inhibition of KDM5A (unknown origin ) by Cellular luciferase reporter assay
Inhibition of KDM5A (unknown origin ) demethylase activity
Assay data:4 Active, 4 Activity ≤ 1 µM, 4 Tested
Inhibition of KDM5A (unknown origin ) by Alphalisa analysis
Assay data:4 Active, 4 Activity ≤ 1 µM, 5 Tested
Inhibition of KDM5A (unknown origin ) by HTMS analysis
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Inhibition of KDM5A (unknown origin ) by Alphascreen assay
Assay data:15 Active, 11 Activity ≤ 1 µM, 16 Tested
Competitive inhibition of KDM5A (unknown origin) in human HeLa cells by TR-FRET assay
Assay data:1 Tested
Competitive inhibition of KDM5A (unknown origin) in human MM1.S cells by TR-FRET assay
Inhibition of N-terminal his6-tagged human KDM5A (1 to 797 residues) expressed in sf9 insect cells incubated for 20 mins by Alphascreen assay
Assay data:7 Active, 2 Activity ≤ 1 µM, 8 Tested
Inhibition of KDM5A (unknown origin) using H3K4me3 as substrate by MSD ELISA analysis
Biochemical KDM5A Inhibition Assay from US Patent US11691968: "Compound having KDM5 inhibitory activity and pharmaceutical use thereof"
Assay data:44 Active, 44 Activity ≤ 1 µM, 44 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Inhibition of KDM5A (unknown origin) in presence of 300 uM 2-OG
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of KDM5A (unknown origin) in presence of 4 uM 2-OG
Inhibition of recombinant HQ5-Halo-tagged KDM5A PHD3 domain (unknown origin) measured by fluorescence polarization assay
Assay data:2 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of KDM5A (unknown origin) measured by AlphaScreen assay
Assay data:3 Active, 3 Activity ≤ 1 µM, 3 Tested
Inhibition of KDM5A (unknown origin) measured by ELISA assay
Inhibition of full-length KDM5A (1 to 1090 residues)(unknown origin) using ARTK(me3)-QTARKSTGGKAPRKQLA-GGK(biotin) as substrate preincubated for 10 mins followed by substrate addition measured after 45 mins by LANCE Ultra assay
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of full-length human KDM5A expressed in recombinant baculovirus expression system using H3K9me3 peptide as substrate incubated for 30 to 45 mins by TR-FRET assay
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