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Reversible inhibition of activated human TG3 using peptidic FRET-quenched probe A101 as substrate by fluorescence based assay relative to control
Assay data:4 Tested
SummaryRelated BioAssays by Target
Inhibition of TG3 (unknown origin) using peptidic FRET quenched probe A101 as substrate and measured by fluorescence-based assay
Assay data:3 Tested
SummaryPubMed CitationRelated BioAssays by Target
Transamidation Assay for Determining Inhibitor Selectivity from US Patent US11472838: "Inhibitors of blood coagulation factor XIII"
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
TG Activity Assays from Article 10.1016/j.chembiol.2015.08.013: "Development of Potent and Selective Tissue Transglutaminase Inhibitors: Their Effect on TG2 Function and Application in Pathological Conditions."
Assay data:27 Active, 14 Activity ≤ 1 µM, 29 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inactivation of activated human TG3 assessed as rate constant of enzyme inactivation using FRET- quenched A101 as substrate by fluorescence assay
Assay data:2 Tested
Irreversible inhibition of human TGase 3 assessed as ratio of Kinact/Ki using Z-Glu(HMC)-Gly-OH as substrate measured at 20 secs interval over 900 secs by fluorimetric assay
Inhibition of human transglutaminase 3 using ((benzyloxy)carbonyl)-L-glutaminyl-L-serine peptide substrate assessed as Kinh/Ki ratio by GDH coupled assay
Assay data:8 Tested
Inhibition of transglutaminase 3
Inhibition of human TGM3
Assay data:1 Tested
Inhibition of thrombin activated human TG3 by fluorescent transamidation assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 69 Tested
Experimentally measured binding affinity data derived from PDB
Assay data:3073 Active, 3073 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
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