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Inhibition of rat somatostatin receptor type 5
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryRelated BioAssays by Target
Inhibition of human somatostatin receptor type 5
Assay data:2 Activity ≤ 1 µM, 2 Tested
Inhibition of human somatostatin receptor type 4
Assay data:1 Active, 3 Activity ≤ 1 µM, 3 Tested
Inhibition of human somatostatin receptor type 3
Assay data:2 Activity ≤ 1 µM, 3 Tested
Inhibition of human somatostatin receptor type 2
Inhibition of human somatostatin receptor type 1
Binding affinity to human somatostatin receptor type 5
Binding affinity to human somatostatin receptor type 4
Binding affinity to human somatostatin receptor type 3
Binding affinity to human somatostatin receptor type 2
Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 1 Tested
Binding affinity to human somatostatin receptor type 1
Assay data:1 Active, 1 Tested
Inhibition of human SSTR2
Assay data:3 Active, 3 Activity ≤ 1 µM, 3 Tested
Agonist activity at rat SST2 receptor
Agonist activity at human SST5 receptor expressed in CHO-K1 cells assessed as inhibition of NKH477-induced intracellular cAMP accumulation incubated for 20 mins by HTRF assay
Assay data:7 Activity ≤ 1 µM, 7 Tested
Agonist activity at human SST4 receptor expressed in CHO-K1 cells assessed as inhibition of NKH477-induced intracellular cAMP accumulation incubated for 20 mins by HTRF assay
Assay data:8 Active, 11 Activity ≤ 1 µM, 12 Tested
Agonist activity at human SST3 receptor expressed in CHO-K1 cells assessed as inhibition of NKH477-induced intracellular cAMP accumulation incubated for 20 mins by HTRF assay
Assay data:1 Active, 7 Activity ≤ 1 µM, 7 Tested
Agonist activity at human SST1 receptor expressed in CHO-K1 cells assessed as inhibition of NKH477-induced intracellular cAMP accumulation incubated for 20 mins by HTRF assay
Agonist activity at human SST2 receptor expressed in CHO-K1 cells assessed as inhibition of NKH477-induced intracellular cAMP accumulation incubated for 20 mins by HTRF assay
Assay data:30 Active, 8 Activity ≤ 1 nM, 30 Activity ≤ 1 µM, 30 Tested
Binding Assay from US Patent US11834435: "SSTR4 agonist salts"
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Displacement of [125I]-Tyr-SRIF 14 from SST5 receptor (unknown origin) expressed in membrane measured after 90 mins by gamma counting analysis
Assay data:2 Active, 33 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
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