Related BioAssays, by Target Similarity (List) for PubChem BioAssay (S - PubChem BioAssay - NCBI

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Select item 19629231.

GPRK5 SGC Tm panel (DSF)

Source:: ChEMBL

Protein Target:: G protein-coupled receptor kinase 5

Assay data:1 Tested

AID:: 1962923

Summary Related BioAssays by Target

Select item 19628192.

GPRK5 SGC Tm panel (DSF)

Source:: ChEMBL

Protein Target:: G protein-coupled receptor kinase 5

Assay data:1 Tested

AID:: 1962819

Summary Related BioAssays by Target

Select item 19627203.

GPRK5 SGC Tm panel (DSF)

Source:: ChEMBL

Protein Target:: G protein-coupled receptor kinase 5

Assay data:1 Tested

AID:: 1962720

Summary Related BioAssays by Target

Select item 19626214.

GPRK5 SGC Tm panel (DSF)

Source:: ChEMBL

Protein Target:: G protein-coupled receptor kinase 5

Assay data:1 Tested

AID:: 1962621

Summary Related BioAssays by Target

Select item 19139795.

Selectivity interaction (KinomeScan (DiscoverX)) EUB0000702a GRK4

Source:: ChEMBL

Protein Target:: G protein-coupled receptor kinase 4

Assay data:1 Tested

AID:: 1913979

Summary Related BioAssays by Target

Select item 19125426.

Thermal Shift Assay. Domain: start/stop: M1-E544

Source:: ChEMBL

Protein Target:: G protein-coupled receptor kinase 5

Assay data:27 Tested

AID:: 1912542

Summary Related BioAssays by Target

Select item 19025717.

Inhibition of human wild type full length GPRK4 (M1 to C578 residues) expressed in bacterial expression system assessed as remaining activity at 1 uM relative to control

Source:: ChEMBL

Protein Target:: G protein-coupled receptor kinase 4

Assay data:1 Tested

AID:: 1902571

Summary PubMed Citation Related BioAssays by Target

Select item 18940598.

Inhibition of GRK6 (unknown origin)

Source:: ChEMBL

Protein Target:: G protein-coupled receptor kinase 6

Assay data:1 Tested

AID:: 1894059

Summary PubMed Citation Related BioAssays by Target

Select item 18940589.

Inhibition of GRK5 (unknown origin)

Source:: ChEMBL

Protein Target:: G protein-coupled receptor kinase 5

Assay data:1 Active, 1 Tested

AID:: 1894058

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 183549310.

GRK4 DiscoveRx kinase panel

Source:: ChEMBL

Protein Target:: G protein-coupled receptor kinase 4

Assay data:1 Tested

AID:: 1835493

Summary Related BioAssays by Target

Select item 183527611.

GPRK5 SGC Tm panel (DSF)

Source:: ChEMBL

Protein Target:: G protein-coupled receptor kinase 5

Assay data:1 Tested

AID:: 1835276

Summary Related BioAssays by Target

Select item 183498212.

GRK6(h) Kinase panel

Source:: ChEMBL

Protein Target:: G protein-coupled receptor kinase 6

Assay data:1 Tested

AID:: 1834982

Summary Related BioAssays by Target

Select item 183498113.

GRK5(h) Kinase panel

Source:: ChEMBL

Protein Target:: G protein-coupled receptor kinase 5

Assay data:1 Tested

AID:: 1834981

Summary Related BioAssays by Target

Select item 183415514.

Inhibition of GRK6 (unknown origin) at 1 uM

Source:: ChEMBL

Protein Target:: G protein-coupled receptor kinase 6

Assay data:1 Tested

AID:: 1834155

Summary PubMed Citation Related BioAssays by Target

Select item 183415415.

Inhibition of GRK5 (unknown origin) at 1 uM

Source:: ChEMBL

Protein Target:: G protein-coupled receptor kinase 5

Assay data:1 Tested

AID:: 1834154

Summary PubMed Citation Related BioAssays by Target

Select item 183415316.

Inhibition of GRK4 (unknown origin) at 1 uM

Source:: ChEMBL

Protein Target:: G protein-coupled receptor kinase 4

Assay data:1 Tested

AID:: 1834153

Summary PubMed Citation Related BioAssays by Target

Select item 181628817.

Inhibition of human recombinant GRK5 assessed as reduction in substrate phosphorylation at 50 to 500 nM using ATP and Ulight-CKKSRGDYMTMQIG (IRS-1) incubated for 60 min by LANCE detection method

Source:: ChEMBL

Protein Target:: G protein-coupled receptor kinase 5

Assay data:1 Tested

AID:: 1816288

Summary PubMed Citation Related BioAssays by Target

Select item 179826718.

TBD from US Patent US10252984: "Inhibiting G protein coupled receptor 6 kinase polypeptides"

Source:: BindingDB

Protein Targets:: G protein-coupled receptor kinase 6; ...
Total:: 1

Assay data:25 Active, 1 Activity ≤ 1 µM, 51 Tested

AID:: 1798267

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 179566319.

Assays for Inhibition of GRKs from US Patent US10023564: "G protein-coupled receptor kinase 2 inhibitors and methods for use of the same"

Source:: BindingDB

Protein Targets:: Beta-adrenergic receptor kinase 1; ...
Total:: 3

Assay data:35 Active, 23 Activity ≤ 1 µM, 39 Tested

AID:: 1795663

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Depositor Related BioAssays by Target

Select item 179411820.

KinomeScan assay: inhibition of GRK4

Source:: ChEMBL

Protein Target:: G protein-coupled receptor kinase 4

Assay data:1 Active, 108 Tested

AID:: 1794118

Summary Compounds, Active Related BioAssays by Target

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Proteins (4)
BioAssays with protein sequences specified as targets

BioActivity

Active Compounds (62)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (1)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (43)
BioAssays with the active concentration of tested reagents less than 1 micromolar

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Confirmatory (77)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations

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Literature Extraction (233)
BioAssays extracted from the literature
Other (79)
BioAssays deposited by other experimentalists

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Related BioAssays, by Target Similarity (List) for PubChem BioAss... (312)
Related BioAssays, by Target Similarity (List) for PubChem BioAssay (Select 1260037)
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PubChem BioAssay
Homo sapiens nucleosome assembly protein 1 like 3 (NAP1L3), RefSeqGene on chromo...
Homo sapiens nucleosome assembly protein 1 like 3 (NAP1L3), RefSeqGene on chromosome X
gi|261862283|ref|NG_013275.1|

Nucleotide
Homo sapiens collagen type VII alpha 1 chain (COL7A1), mRNA
Homo sapiens collagen type VII alpha 1 chain (COL7A1), mRNA
gi|1812585486|ref|NM_000094.4|

Nucleotide
AU014937 Mouse two-cell stage embryo cDNA Mus musculus cDNA clone J0704H04 3', m...
AU014937 Mouse two-cell stage embryo cDNA Mus musculus cDNA clone J0704H04 3', mRNA sequence
gi|3369728|gnl|dbEST|1816330|dbj|AU 7.1|

Nucleotide

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