BioAssay by Target (List) for Gene (Select 2444) - PubChem BioAssay - NCBI

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Select item 19138111.

Selectivity interaction (Z?-LYTE assay (SelectScreen Invitrogen)) EUB0000690a FRK

Source:: ChEMBL

Protein Target:: Tyrosine-protein kinase FRK

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1913811

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 19137252.

Selectivity interaction (33P-ATP and filter-binding assay (Reaction Biology)) EUB0000646a FRK

Source:: ChEMBL

Protein Target:: Tyrosine-protein kinase FRK

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1913725

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 19135783.

Selectivity interaction (KinomeScan (DiscoverX)) EUB0000147b FRK

Source:: ChEMBL

Protein Target:: Tyrosine-protein kinase FRK

Assay data:1 Tested

AID:: 1913578

Summary Related BioAssays by Target

Select item 19135204.

Selectivity interaction (Ambit kinome screening platform (Ambit phage-based competition binding assay)) EUB0000624a FRK

Source:: ChEMBL

Protein Target:: Tyrosine-protein kinase FRK

Assay data:1 Tested

AID:: 1913520

Summary Related BioAssays by Target

Select item 18355335.

FRK DiscoveRx kinase panel

Source:: ChEMBL

Protein Target:: Tyrosine-protein kinase FRK

Assay data:1 Tested

AID:: 1835533

Summary Related BioAssays by Target

Select item 18351336.

PTK5(h) Kinase panel

Source:: ChEMBL

Protein Target:: Tyrosine-protein kinase FRK

Assay data:1 Tested

AID:: 1835133

Summary Related BioAssays by Target

Select item 18341467.

Inhibition of FRK (unknown origin) at 1 uM

Source:: ChEMBL

Protein Target:: Tyrosine-protein kinase FRK

Assay data:1 Tested

AID:: 1834146

Summary PubMed Citation Related BioAssays by Target

Select item 18224588.

Inhibition of human PTK5 in presence of ATP by radiometric assay

Source:: ChEMBL

Protein Target:: Tyrosine-protein kinase FRK

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1822458

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 18050459.

Radioisotope Filter Binding Assay from US Patent US10844038: "1,2-dithiolane compounds useful in neuroprotection, autoimmune and cancer diseases and conditions"

Source:: BindingDB

Protein Targets:: Aurora kinase A; ...
Total:: 20

Assay data:12 Active, 9 Activity ≤ 1 µM, 12 Tested

AID:: 1805045

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Depositor Related BioAssays by Target

Select item 179873910.

Kinase Screening Assay from US Patent US10294227: "Compounds"

Source:: BindingDB

Protein Targets:: Mast/stem cell growth factor receptor Kit; ...
Total:: 15

Assay data:20 Active, 21 Activity ≤ 1 µM, 21 Tested

AID:: 1798739

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 179857011.

Z-LYTE Enzymatic Kinase Assay from Article 10.1073/pnas.0711741105: "Discovery of a selective inhibitor of oncogenic B-Raf kinase with potent antimelanoma activity."

Source:: BindingDB

Protein Targets:: Protein-tyrosine kinase 6; ...
Total:: 4

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1798570

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Depositor Related BioAssays by Target

Select item 179840312.

Kinase Inhibition Assays from US Patent US10266537: "3-acetylenyl-pyrazole-pyrimidine derivative, and preparation method therefor and uses thereof"

Source:: BindingDB

Protein Targets:: Angiopoietin-1 receptor; ...
Total:: 42

Assay data:27 Active, 4 Activity ≤ 1 nM, 26 Activity ≤ 1 µM, 27 Tested

AID:: 1798403

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 179411113.

KinomeScan assay: inhibition of FRK

Source:: ChEMBL

Protein Target:: Tyrosine-protein kinase FRK

Assay data:108 Tested

AID:: 1794111

Summary Related BioAssays by Target

Select item 179368014.

FRK(FRK1LGF1) Takeda global kinase panel

Source:: ChEMBL

Protein Target:: Tyrosine-protein kinase FRK

Assay data:1 Activity ≤ 1 µM, 1 Tested

AID:: 1793680

Summary Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 179338915.

FRK(FRK1LGF1) Takeda global kinase panel

Source:: ChEMBL

Protein Target:: Tyrosine-protein kinase FRK

Assay data:1 Activity ≤ 1 µM, 1 Tested

AID:: 1793389

Summary Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 179309516.

FRK(FRK1LGF1) Takeda global kinase panel

Source:: ChEMBL

Protein Target:: Tyrosine-protein kinase FRK

Assay data:1 Activity ≤ 1 µM, 1 Tested

AID:: 1793095

Summary Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 179282917.

PTK5(h) Eurofins kinase panel

Source:: ChEMBL

Protein Target:: Tyrosine-protein kinase FRK

Assay data:1 Tested

AID:: 1792829

Summary Related BioAssays by Target

Select item 179230018.

FRK ProQinase selectivity panel

Source:: ChEMBL

Protein Target:: Tyrosine-protein kinase FRK

Assay data:1 Tested

AID:: 1792300

Summary Related BioAssays by Target

Select item 179101619.

FRK (PTK5) Kinase screen

Source:: ChEMBL

Protein Target:: Tyrosine-protein kinase FRK

Assay data:1 Tested

AID:: 1791016

Summary Related BioAssays by Target

Select item 179019520.

FRK Invitrogen selectivity data (BI)

Source:: ChEMBL

Protein Target:: Tyrosine-protein kinase FRK

Assay data:1 Tested

AID:: 1790195

Summary Related BioAssays by Target

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Target

Proteins (3)
BioAssays with protein sequences specified as targets
RNAi Target, Active (10)
BioAssays with gene sequences specified as RNAi targets and the activity is active

BioActivity

Active Compounds (43)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (6)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (40)
BioAssays with the active concentration of tested reagents less than 1 micromolar

Experiment Type

Summary (1)
BioAssays summarizing information from multiple assays for validated chemical probes or small molecule leads
Confirmatory (43)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations
Primary Screening (40)
Primary high-throughput BioAssays where the activity outcome is based on percentage inhibition from a single dose
Chemical Screens (172)
BioAssays reporting BioActivity of chemical reagents
RNAi Screens (46)
BioAssays reporting BioActivity of RNAi reagents

Assay Project (1)
BioAssays organized into assay projects based on linkage to Summary assays. Click an project below to retrieve the bioassay list for the project. Click 'All Assay Projects' to retrieve all assay projects represented by Summary assays.

Depositor Category

Literature Extraction (139)
BioAssays extracted from the literature
NIH MLP (2)
BioAssays deposited by the NIH Molecular Libraries Program
Other (76)
BioAssays deposited by other experimentalists

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