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Summary
Selectivity interaction (BROMOscan? panel (DiscoverX)) EUB0000256b BPTF
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Selectivity interaction (Bromodomain panel (DSF assay)) EUB0000253b BPTF
Assay data:1 Tested
SummaryRelated BioAssays by Target
Selectivity interaction (AlphaScreen) EUB0000253b BPTF
Selectivity interaction (Bromodomain panel (DSF assay)) EUB0000201c BPTF
Affinity Biochemical interaction (BioLayer Interferometry assay (BLI)) EUB0000254b BPTF
Assay data:1 Active, 1 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
Affinity Biochemical interaction (BioLayer Interferometry assay (BLI)) EUB0000253b BPTF
Affinity On-target Cellular interaction (NanoBRET assay (HEK293T cells)) EUB0000254b BPTF
Affinity On-target Cellular interaction (NanoBRET assay (HEK293T cells)) EUB0000253b BPTF
Cellular target engagement assay with: BPTFBRD
Binding affinity to N-terminal His-TEV-tagged human BPTF-BD2 transfected in Escherichia coli BL21 (DE3) assessed as thermal stabilization by measuring change in melting temperature at 100 uM by SYPRO orange dye based differential scanning fluorimetry analysis
SummaryPubMed CitationRelated BioAssays by Target
Binding affinity to human FALZ bromodomain by BROMOscan method
Assay data:1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Binding affinity to human FALZ bromodomain assessed as residual activity at 300 nM by BROMOscan method relative to control
FALZ DiscoverX BROMOscan
Binding affinity to BPTF (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by SPR analysis
Assay data:3 Active, 1 Activity ≤ 1 µM, 3 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Binding affinity to BPTF (unknown origin)
Assay data:2 Active, 2 Activity ≤ 1 µM, 3 Tested
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