BioAssay by Target (List) for Gene (Select 1551) - PubChem BioAssay - NCBI

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Select item 19184321.

Inhibition of CYP450 (unknown origin)

Source:: ChEMBL

Protein Targets:: Cytochrome P450 1A1; ...
Total:: 29

Assay data:1 Tested

AID:: 1918432

Summary PubMed Citation Related BioAssays by Target

Select item 18733342.

Inhibition of CYP450 (unknown origin)

Source:: ChEMBL

Protein Targets:: Cytochrome P450 1A1; ...
Total:: 29

Assay data:2 Tested

AID:: 1873334

Summary PubMed Citation Related BioAssays by Target

Select item 18709853.

Metabolic stability of the compound in human liver microsomes assessed as CYP450-mediated metabolism by measuring parent compound remaining at 0.5 uM measured after 10 mins in presence of NADPH by LC-MS/MS analysis

Source:: ChEMBL

Protein Targets:: Cytochrome P450 1A1; ...
Total:: 29

Assay data:1 Tested

AID:: 1870985

Summary PubMed Citation Related BioAssays by Target

Select item 18687084.

Metabolic stability in human liver microsomes S9 fraction assessed as CYP450-mediated metabolism by measuring parent compound remaining measured after 60 mins in presence of NADPH

Source:: ChEMBL

Protein Targets:: Cytochrome P450 1A1; ...
Total:: 29

Assay data:2 Tested

AID:: 1868708

Summary PubMed Citation Related BioAssays by Target

Select item 18687075.

Metabolic stability in human liver microsomes S9 fraction assessed as CYP450-mediated metabolism by measuring parent compound remaining measured after 30 mins in presence of NADPH

Source:: ChEMBL

Protein Targets:: Cytochrome P450 1A1; ...
Total:: 29

Assay data:2 Tested

AID:: 1868707

Summary PubMed Citation Related BioAssays by Target

Select item 18687066.

Metabolic stability in human liver microsomes S9 fraction assessed as CYP450-mediated metabolism by measuring parent compound remaining measured after 15 mins in presence of NADPH

Source:: ChEMBL

Protein Targets:: Cytochrome P450 1A1; ...
Total:: 29

Assay data:2 Tested

AID:: 1868706

Summary PubMed Citation Related BioAssays by Target

Select item 18614027.

Induction of CYP450 (unknown origin)

Source:: ChEMBL

Protein Targets:: Cytochrome P450 1A1; ...
Total:: 29

Assay data:1 Tested

AID:: 1861402

Summary PubMed Citation Related BioAssays by Target

Select item 18614018.

Inhibition of CYP450 (unknown origin)

Source:: ChEMBL

Protein Targets:: Cytochrome P450 1A1; ...
Total:: 29

Assay data:1 Tested

AID:: 1861401

Summary PubMed Citation Related BioAssays by Target

Select item 18603699.

Inhibition of CYP450 in human HCT-116 cells assessed as 20-HETE formation in presence of arachidonic acid incubated for 15 mins by multi-enzyme assay based LC-MS/MS analysis

Source:: ChEMBL

Protein Targets:: Cytochrome P450 1A1; ...
Total:: 29

Assay data:1 Active, 1 Tested

AID:: 1860369

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 186036810.

Inhibition of CYP450 in human HCT-116 cells assessed as 20-HETE formation in presence of arachidonic acid incubated for 15 mins by multi-enzyme assay based LC-MS/MS analysis relative to control

Source:: ChEMBL

Protein Targets:: Cytochrome P450 1A1; ...
Total:: 29

Assay data:1 Active, 1 Tested

AID:: 1860368

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 186035711.

Inhibition of CYP450 in human liver microsomes assessed as inhibition of 20-HETE formation in presence of arachidonic acid and NADPH by multi-enzyme assay based LC-MS/MS analysis relative to control

Source:: ChEMBL

Protein Targets:: Cytochrome P450 1A1; ...
Total:: 29

Assay data:1 Active, 1 Tested

AID:: 1860357

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 186035612.

Inhibition of CYP450 in human liver microsomes assessed as inhibition of 20-HETE formation in presence of arachidonic acid and NADPH by multi-enzyme assay based LC-MS/MS analysis

Source:: ChEMBL

Protein Targets:: Cytochrome P450 1A1; ...
Total:: 29

Assay data:1 Active, 1 Tested

AID:: 1860356

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 186035413.

Inhibition of CYP450 in human liver microsomes assessed as inhibition of EpETrE formation at 10 uM in presence of arachidonic acid and NADPH by multi-enzyme assay based LC-MS/MS analysis relative to control

Source:: ChEMBL

Protein Targets:: Cytochrome P450 1A1; ...
Total:: 29

Assay data:31 Tested

AID:: 1860354

Summary PubMed Citation Related BioAssays by Target

Select item 186035314.

Inhibition of CYP450 in human liver microsomes assessed as inhibition of 20-HETE formation at 10 uM in presence of arachidonic acid and NADPH by multi-enzyme assay based LC-MS/MS analysis relative to control

Source:: ChEMBL

Protein Targets:: Cytochrome P450 1A1; ...
Total:: 29

Assay data:31 Tested

AID:: 1860353

Summary PubMed Citation Related BioAssays by Target

Select item 185711415.

Metabolic stability assessed as P450 (unknown origin)-mediated biotransformation assessed as compound remaining measured after 120 mins

Source:: ChEMBL

Protein Targets:: Cytochrome P450 1A1; ...
Total:: 29

Assay data:2 Tested

AID:: 1857114

Summary PubMed Citation Related BioAssays by Target

Select item 185711316.

Metabolic stability assessed as P450 (unknown origin)-mediated biotransformation assessed as compound remaining measured after 15 mins

Source:: ChEMBL

Protein Targets:: Cytochrome P450 1A1; ...
Total:: 29

Assay data:1 Tested

AID:: 1857113

Summary PubMed Citation Related BioAssays by Target

Select item 185000617.

Drug metabolism in human hepatocytes assessed as fraction of Cyp mediated oxidative metabolism in presence of NADPH

Source:: ChEMBL

Protein Targets:: Cytochrome P450 1A1; ...
Total:: 29

Assay data:2 Tested

AID:: 1850006

Summary PubMed Citation Related BioAssays by Target

Select item 184970718.

Inhibition of CYP450 (unknown origin)

Source:: ChEMBL

Protein Targets:: Cytochrome P450 1A1; ...
Total:: 29

Assay data:3 Tested

AID:: 1849707

Summary PubMed Citation Related BioAssays by Target

Select item 183012719.

Inhibition of CYP (unknown origin)

Source:: ChEMBL

Protein Targets:: Cytochrome P450 1A1; ...
Total:: 29

Assay data:1 Tested

AID:: 1830127

Summary PubMed Citation Related BioAssays by Target

Select item 183012620.

Induction of CYP (unknown origin)

Source:: ChEMBL

Protein Targets:: Cytochrome P450 1A1; ...
Total:: 29

Assay data:1 Tested

AID:: 1830126

Summary PubMed Citation Related BioAssays by Target

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Target

RNAi Target, Active (6)
BioAssays with gene sequences specified as RNAi targets and the activity is active

BioActivity

Active Compounds (32)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 µM (10)
BioAssays with the active concentration of tested reagents less than 1 micromolar

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BioAssays summarizing information from multiple assays for validated chemical probes or small molecule leads
Confirmatory (60)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations
Primary Screening (8)
Primary high-throughput BioAssays where the activity outcome is based on percentage inhibition from a single dose
Chemical Screens (212)
BioAssays reporting BioActivity of chemical reagents
RNAi Screens (12)
BioAssays reporting BioActivity of RNAi reagents

Assay Project (1)
BioAssays organized into assay projects based on linkage to Summary assays. Click an project below to retrieve the bioassay list for the project. Click 'All Assay Projects' to retrieve all assay projects represented by Summary assays.

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Literature Extraction (209)
BioAssays extracted from the literature
NIH MLP (1)
BioAssays deposited by the NIH Molecular Libraries Program
Other (14)
BioAssays deposited by other experimentalists

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